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Relugolix, MedChemExpress

Product Code. 16467058
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Product Code. 16467058 Supplier Medchem Express Supplier No. HY16474

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Description

MedChemExpress Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.

Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.

Specifications

Chemical Name or Material Relugolix
CAS 737789-87-6
Color Off-White
Purity Grade Notes Research
Molecular Formula C29H27F2N7O5S
Quantity 10 mg
Synonym TAK-385
Solubility Information DMSO : 100 mg/mL (160.35 mM; Need ultrasonic)
SMILES O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1
Molecular Weight (g/mol) 623.63
Formula Weight 623.63
Percent Purity 99.51%
Grade Research
Physical Form Powder
For Use With (Application) Cancer-programmed cell death
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Research purposes only

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