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MSG 606, Tocris Bioscience™

Product Code. 30000954
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1 mg
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Product Code. 30000954 Supplier Tocris Bioscience Supplier No. 5954/1

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Description

Potent human MC1 receptor antagonist; also MC3 and MC5 partial agonist

Potent human MC1 receptor antagonist (IC50 = 17 nM). Also partial agonist at human MC3 and MC5 receptors (EC50 values are 59 and 1300 nM, respectively). Exhibits binding affinity for A375 melanoma cells in vitro. Reverses morphine-induced hyperalgesia in female mice, with no effect in male mice. γMSH analog.
TRUSTED_SUSTAINABILITY

Specifications

CAS 1416983-77-1
Molecular Formula C62H82N20O13S
Linear Formula C62H82N20O13S
Quantity 1 mg
Solubility Information Soluble to 1mg/mL in water
InChI Key QJBNFEXQHBDMQM-VTWSTLNFSA-N
SMILES C1CC(=O)NCC(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(CSC1)C(=O)NC(CC(=O)O)C(=O)NC(CCCN=C(N)N)C(=O)NC(CC2=CC=CC=C2)C(=O)NCC(=O)N)CC3=CNC4=CC=CC=C43)CCCN=C(N)N)CC5=CC=CC=C5)CC6=CN=CN6
IUPAC Name (3S)-4-[[(2S)-1-[[(2S)-1-[(2-amino-2-oxoethyl)amino]-1-oxo-3-phenylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-[[(3R,6S,9S,12S,15S)-12-benzyl-9-[3-(diaminomethylideneamino)propyl]-15-(1H-imidazol-5-ylmethyl)-6-(1H-indol-3-ylme
Molecular Weight (g/mol) 1347.525
PubChem CID 122177131
Formula Weight 1347.51
Percent Purity 0.95
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