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Ilginatinib maleate, MedChemExpress

Product Code. 16447828
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Product Code. 16447828 Supplier Medchem Express Supplier No. HY19631

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Description

MedChemExpress Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable JAK2 inhibitor, with an IC50 of 0.72 nM, 46-, 54-, and 31-fold selectivity for JAK2 over JAK1 (IC50, 33 nM), JAK3 (IC50, 39 nM), and Tyk2 (IC50, 22 nM).

Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable JAK2 inhibitor, with an IC50 of 0.72 nM, 46-, 54-, and 31-fold selectivity for JAK2 over JAK1 (IC50, 33 nM), JAK3 (IC50, 39 nM), and Tyk2 (IC50, 22 nM).

Specifications

Chemical Name or Material Ilginatinib maleate
CAS 1354799-87-3
Color Light Yellow
Purity Grade Notes Research
Molecular Formula C25H24FN7O4
Quantity 10 mg
Synonym NS-018 maleate
Solubility Information DMSO : ≥ 30 mg/mL (59.35 mM) ∣H2O : 1 mg/mL (1.98 mM; Need ultrasonic)
SMILES CN1N=CC(C2=CC(N[C@H](C3=CC=C(F)C=C3)C)=NC(NC4=NC=CN=C4)=C2)=C1.O=C(O)/C=C\C(O)=O
Molecular Weight (g/mol) 505.5
Formula Weight 505.5
Percent Purity 97.04%
Grade Research
Physical Form Solid
For Use With (Application) Cancer-Kinase/protease
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Research purposes only

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